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阿片受体拮抗药
释义
阿片受体拮抗药
Encyclopedia
医学
阿片受体拮抗药
释
opioid receptor antagonist
阿片受体拮抗药
化学结构与吗啡相似,对阿片受体(μ、κ、δ)有很好的亲和力,但无内在活性,不产生激动效应,可置换与这些受体结合的阿片类镇痛药物,从而产生拮抗效应的药物。
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更新时间:2025/4/25 21:49:02